| Codeine 30 | 🇨🇦Canada | 30 MG | Tablet | Marketed | Laboratoire Riva INC. |
| Codeine 15 | 🇨🇦Canada | 15 MG | Tablet | Not marketed | Laboratoire Riva INC. |
| Codeine Phosphate Syrup | 🇨🇦Canada | 25 MG / 5 ML | Syrup | Marketed | Laboratoire Atlas INC |
| Codeine Contin 50MG Controlled Release Tab | 🇨🇦Canada | 50 MG | Tablet (Extended-Release) | Marketed | Purdue Pharma |
| Codeine Contin 100MG Controlled Release Tab | 🇨🇦Canada | 100 MG | Tablet (Extended-Release) | Marketed | Purdue Pharma |
| Codeine Contin 150MG Controlled Release Tab | 🇨🇦Canada | 150 MG | Tablet (Extended-Release) | Marketed | Purdue Pharma |
| Codeine Contin 200MG Controlled Release Tab | 🇨🇦Canada | 200 MG | Tablet (Extended-Release) | Marketed | Purdue Pharma |
| Teva-Codeine | 🇨🇦Canada | 30 MG | Tablet | Marketed | Teva Canada Limited |
| Teva-Codeine | 🇨🇦Canada | 15 MG | Tablet | Marketed | Teva Canada Limited |
| Codeine Tab 15MG | 🇨🇦Canada | 15 MG | Tablet | Cancelled | Rougier Pharma Division of Ratiopharm INC |
| Codeine Tab 30MG | 🇨🇦Canada | 30 MG | Tablet | Cancelled | Rougier Pharma Division of Ratiopharm INC |
| Linctus Codeine Blanc | 🇨🇦Canada | 10 MG / 5 ML | Solution | Marketed | Laboratoire Atlas INC |
| Mersyndol with CodeineCombination | 🇨🇦Canada | 325 MG + 8 MG + 5 MG | Tablet | Marketed | Sanofi-Aventis Canada INC |
| Calmylin Pse with CodeineCombination | 🇨🇦Canada | 3.3 MG / 5 ML + 100 MG / 5 ML + 30 MG / 5 ML | Syrup | Marketed | Teva Canada Limited |
| Cough Syrup with CodeineCombination | 🇨🇦Canada | 3.3 MG / 5 ML + 100 MG / 5 ML + 30 MG / 5 ML | Syrup | Authorised | Cellchem Pharmaceuticals INC. |
| Damylin with Codeine SyrupCombination | 🇨🇦Canada | 125 MG / 5 ML + 3.3 MG / 5 ML + 12.5 MG / 5 ML | Syrup | Marketed | Laboratoire Riva INC. |
| Codeine Phosphate Syrup | 🇨🇦Canada | 5 MG / ML | Syrup | Cancelled | D.C. Labs Limited |
| Damylin Avec Codeine SiropCombination | 🇨🇦Canada | 125 MG / 5 ML + 3.3 MG / 5 ML + 12.5 MG / 5 ML | Syrup | Authorised | Laboratoire Atlas INC |
| Acetaminophen with Codeine - CapletCombination | 🇨🇦Canada | 300 MG + 15 MG + 8 MG | Tablet | Marketed | Teva Canada Limited |
| Codeine Phosphate Tab 15MG | 🇨🇦Canada | 15 MG | Tablet | Cancelled | D.C. Labs Limited |
| Codeine Phosphate Tab 30MG | 🇨🇦Canada | 30 MG | Tablet | Cancelled | D.C. Labs Limited |
| Codeine Phosphate Tab 60MG | 🇨🇦Canada | 60 MG | Tablet | Cancelled | D.C. Labs Limited |
| PMS-Acetaminophen with Codeine ElixirCombination | 🇨🇦Canada | 160 MG / 5 ML + 8 MG / 5 ML | Elixir | Marketed | Pharmascience INC |
| Cough Syrup with CodeineCombination | 🇨🇦Canada | 3.3 MG / 5 ML + 100 MG / 5 ML + 30 MG / 5 ML | Syrup | Not marketed | Jamp Pharma Corporation |
| Acetaminophen 300MG, Caffeine & CodeineCombination | 🇨🇦Canada | 300 MG + 15 MG + 8 MG | Tablet | Authorised | Tanta Pharmaceuticals INC |