| Caffeine | 🇨🇦Canada | 200 MG | Tablet | Cancelled | Added Dimensions |
| Caffeine Citrate | 🇺🇸United States | 30MG BASE/3ML | solution | Marketed | Fresenius Kabi USA |
| Caffeine Citrate | 🇺🇸United States | 30MG BASE/3ML | solution | Marketed | Exela Pharma |
| Caffeine 1508 | 🇺🇸United States | | | Status unknown | |
| Caffeine Citrate Injection USP | 🇨🇦Canada | 20 MG / ML | Solution | Marketed | Omega Laboratories Limited |
| Caffeine Citrate Oral Solution USP | 🇨🇦Canada | 20 MG / ML | Solution | Marketed | Omega Laboratories Limited |
| Caffeine and Sodium BenzoateCombination | 🇺🇸United States | | | Status unknown | |
| Butalbital, Aspirin and CaffeineCombination | 🇺🇸United States | 325MG; 50MG; 40MG, 500MG; 50MG; 40MG | capsule | Marketed | MPP Pharma |
| Ergotamine Tartrate and CaffeineCombination | 🇺🇸United States | 100MG; 1MG | tablet | Marketed | Hikma Intl Pharms |
| Acetaminophen, Aspirin and CaffeineCombination | 🇺🇸United States | 250MG; 250MG; 65MG | tablet | Marketed | Granules |
| Butalbital, Acetaminophen and CaffeineCombination | 🇺🇸United States | 300MG; 50MG; 40MG, 325MG; 50MG; 40MG, 325MG; 50MG; 40MG **Federal Register determination that product was not discontinued or withdrawn for safety or effectiveness reasons** … | capsule | Marketed | Gilbert Labs |
| Butalbital, Acetaminophen and CaffeineCombination | 🇺🇸United States | 325MG/15ML; 50MG/15ML; 40MG/15ML | solution | Marketed | Genus |
| Butalbital, Acetaminophen and CaffeineCombination | 🇺🇸United States | 325MG; 50MG; 40MG, 500MG; 50MG; 40MG, 750MG; 50MG; 40MG | tablet | Marketed | Quagen |
| Cafcit | 🇺🇸United States | 30MG BASE/3ML | solution | Marketed | Hikma |
| Butalbital, Aspirin, Caffeine, and Codeine PhosphateCombination | 🇺🇸United States | 325MG; 50MG; 40MG; 30MG | capsule | Marketed | Stevens J |
| Butalbital, Acetaminophen, Caffeine and Codeine PhosphateCombination | 🇺🇸United States | 300MG; 50MG; 40MG; 30MG, 325MG; 50MG; 40MG; 30MG | capsule | Marketed | LGM Pharma |
| Butalbital; Acetaminophen; Caffeine; CodeineCombination | 🇺🇸United States | 40MG/30MG | Capsule | Marketed | Able |
| CAFFEINE CITRATE 10 mg/ml Solution For Injection | 🇸🇦Saudi Arabia | | | Authorised | Macarthys Laboratories Limited T\A Martindale Pharma |
| Cafcit | 🇺🇸United States | 30MG BASE/3ML (EQ 10MG BASE/ML) **Federal Register determination that product was not discontinued or withdrawn for safety or effectiveness reasons** | solution | Not marketed | Hikma |
| Apo-Butalbital-Acetylsalicylic Acid-CaffeineCombination | 🇨🇦Canada | 330 MG + 50 MG + 40 MG | Capsule | Marketed | Apotex INC |
| Acetaminophen 300MG, Caffeine & CodeineCombination | 🇨🇦Canada | 300 MG + 15 MG + 8 MG | Tablet | Authorised | Tanta Pharmaceuticals INC |
| Butalbital, Aspirin and CaffeineCombination | 🇺🇸United States | 325MG; 50MG; 40MG, 325MG; 50MG; 40MG **Federal Register determination that product was not discontinued or withdrawn for safety or effectiveness reasons** | tablet | Not marketed | Quantum Pharmics |
| Acetaminophen 325 MG Caffeine and CodeineCombination | 🇨🇦Canada | 325 MG + 15 MG + 8 MG | Tablet | Authorised | Tanta Pharmaceuticals INC |
| Acetaminophen, Caffeine and Codeine Phosphate TabletsCombination | 🇨🇦Canada | 300 MG + 15 MG + 8 MG | Tablet | Marketed | Laboratoire Riva INC. |
| Apo-Butalbital-Acetylsalicylic Acid-Caffeine-Codeine-C 1/2Combination | 🇨🇦Canada | 330 MG + 50 MG + 40 MG + 30 MG | Capsule | Marketed | Apotex INC |