| Caffeine Citrate | 🇺🇸United States | 30MG BASE/3ML | solution | Marketed | Fresenius Kabi USA |
| Caffeine Citrate | 🇺🇸United States | 30MG BASE/3ML | solution | Marketed | Exela Pharma |
| Caffeine 1508 | 🇺🇸United States | | | Status unknown | |
| Caffeine and Sodium BenzoateCombination | 🇺🇸United States | | | Status unknown | |
| Butalbital, Aspirin and CaffeineCombination | 🇺🇸United States | 325MG; 50MG; 40MG, 500MG; 50MG; 40MG | capsule | Marketed | MPP Pharma |
| Ergotamine Tartrate and CaffeineCombination | 🇺🇸United States | 100MG; 1MG | tablet | Marketed | Hikma Intl Pharms |
| Acetaminophen, Aspirin and CaffeineCombination | 🇺🇸United States | 250MG; 250MG; 65MG | tablet | Marketed | Granules |
| Butalbital, Acetaminophen and CaffeineCombination | 🇺🇸United States | 300MG; 50MG; 40MG, 325MG; 50MG; 40MG, 325MG; 50MG; 40MG **Federal Register determination that product was not discontinued or withdrawn for safety or effectiveness reasons** … | capsule | Marketed | Gilbert Labs |
| Butalbital, Acetaminophen and CaffeineCombination | 🇺🇸United States | 325MG/15ML; 50MG/15ML; 40MG/15ML | solution | Marketed | Genus |
| Butalbital, Acetaminophen and CaffeineCombination | 🇺🇸United States | 325MG; 50MG; 40MG, 500MG; 50MG; 40MG, 750MG; 50MG; 40MG | tablet | Marketed | Quagen |
| Cafcit | 🇺🇸United States | 30MG BASE/3ML | solution | Marketed | Hikma |
| Butalbital, Aspirin, Caffeine, and Codeine PhosphateCombination | 🇺🇸United States | 325MG; 50MG; 40MG; 30MG | capsule | Marketed | Stevens J |
| Butalbital, Acetaminophen, Caffeine and Codeine PhosphateCombination | 🇺🇸United States | 300MG; 50MG; 40MG; 30MG, 325MG; 50MG; 40MG; 30MG | capsule | Marketed | LGM Pharma |
| Butalbital; Acetaminophen; Caffeine; CodeineCombination | 🇺🇸United States | 40MG/30MG | Capsule | Marketed | Able |
| Cafcit | 🇺🇸United States | 30MG BASE/3ML (EQ 10MG BASE/ML) **Federal Register determination that product was not discontinued or withdrawn for safety or effectiveness reasons** | solution | Not marketed | Hikma |
| Butalbital, Aspirin and CaffeineCombination | 🇺🇸United States | 325MG; 50MG; 40MG, 325MG; 50MG; 40MG **Federal Register determination that product was not discontinued or withdrawn for safety or effectiveness reasons** | tablet | Not marketed | Quantum Pharmics |
| Phrenilin with Caffeine and CodeineCombination | 🇺🇸United States | 325MG; 50MG; 40MG; 30MG | capsule | Not marketed | Valeant |
| MigergotCombination | 🇺🇸United States | 100MG; 2MG | suppository | Marketed | Cosette |
| Pain Relief Caffeine and HempCombination | 🇺🇸United States | | | Status unknown | |
| Orphenadrine Citrate, Aspirin, and CaffeineCombination | 🇺🇸United States | 385MG; 30MG; 25MG, 770MG; 60MG; 50MG | tablet | Not marketed | Sandoz |
| CafergotCombination | 🇺🇸United States | 100MG; 1MG | tablet | Not marketed | Novartis |
| CafergotCombination | 🇺🇸United States | 100MG; 2MG **Federal Register determination that product was not discontinued or withdrawn for safety or effectiveness reasons** | suppository | Not marketed | Novartis |
| Caffeine Mix 1003 | 🇺🇸United States | | | Status unknown | |
| Propoxyphene Hydrochloride W/ Aspirin and CaffeineCombination | 🇺🇸United States | 389MG; 32.4MG; 65MG | capsule | Not marketed | Watson Labs |
| Acetaminophen, Caffeine and Dihydrocodeine BitartrateCombination | 🇺🇸United States | 325MG; 30MG; 16MG | tablet | Not marketed | Pharmobedient |