| Sitagliptin | 🇺🇸United States | 100MG, 25MG, 50MG | tablet | Tentative approval | Sciegen Pharmaceuticals INC |
| Sitagliptin | 🇺🇸United States | 100MG, 25MG, 50MG | tablet | Tentative approval | Laurus Labs LTD |
| Sitagliptin | 🇺🇸United States | 100MG, 25MG, 50MG | tablet | Tentative approval | Mankind Pharma LTD |
| Sitagliptin | 🇺🇸United States | 100MG, 50MG | tablet | Tentative approval | Fosun Wanbang (Jiangsu) Pharmaceutical Group Co., |
| Sitagliptin Phosphate | 🇺🇸United States | 100MG, 100MG BASE, 25MG … | tablet | Marketed | Alkem Labs LTD |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 1GM; 50MG BASE, 500MG; 50MG BASE | tablet | Marketed | Apotex |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 1GM; 100MG BASE, 1GM; 50MG BASE, 500MG; 50MG BASE | tablet, extended release | Marketed | PH Health |
| Sitagliptin Phosphate | 🇺🇸United States | 100MG, 25MG, 50MG | tablet | Tentative approval | DR Reddys Labs LTD |
| Sitagliptin and Metformin HCLCombination | 🇺🇸United States | 1000MG, 1000MG ER TABLET, 100MG BASE TABLET … | tablet | Tentative approval | Mankind Pharma LTD |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 1000MG, 50MG | tablet | Tentative approval | Ajanta Pharma LTD |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 1000MG, 100MG, 100MG BASE TABLET … | tablet, extended release | Tentative approval | Apotex INC |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 100MG, 500MG, 50MG | tablet | Tentative approval | MSN Laboratories Private LTD |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 100MG, 500MG, 50MG | tablet, extended release | Tentative approval | Zhejiang Jiuzhou Biopharma Co., LTD. |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 100MG, 500MG, 50MG | tablet, extended release | Tentative approval | Sinotherapeutics INC |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 1000MG, 500MG | tablet | Tentative approval | Aurobindo Pharma Limited |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 500MG, 50MG | tablet, coated | Tentative approval | MSN Laboratories Private LTD |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 500MG, 50MG | tablet | Tentative approval | Inventia Healthcare Limited |
| Sitagliptin and Metformin HydrochlorideCombination | 🇺🇸United States | 50MG/1000MG | tablet | Tentative approval | Ajanta Pharma LTD |
| Sitagliptin Phosphate; Metformin HydrochlorideCombination | 🇺🇸United States | 50MG; 1000MG, 50MG; 500MG | tablet | Tentative approval | Watson Labs INC |
| Sitagliptin Phosphate; Metformin HydrochlorideCombination | 🇺🇸United States | 100MG; 1000MG, 50MG; 1000MG, 50MG; 500MG | tablet, extended release | Tentative approval | Teva Pharms USA INC |
| Sitagliptin Phosphate and Metformin HydrochlorideCombination | 🇺🇸United States | 1000MG, 500MG, 50MG | tablet | Tentative approval | Prinston Pharmaceutical INC |
| Januvia | 🇺🇸United States | 100MG BASE, 25MG BASE, 50MG BASE | tablet | Marketed | MSD |
| Zituvio | 🇺🇸United States | 100MG, 25MG, 50MG | tablet | Marketed | Zydus Lifesciences |
| Brynovin | 🇺🇸United States | 25MG BASE/ML | solution | Marketed | Azurity |
| Metformin Hydrochloride and Sitagliptin PhosphateCombination | 🇺🇸United States | 50MG/500MG; 50MG/1000MG | tablet | Tentative approval | Zydus Pharms USA INC |